中文名称

APD356 | Belviq;?8-氯-2,3,4,5-四氢-1R-甲基-1H-3-苯并ze庚因，一盐酸盐

英文名字

APD356|Belviq; 8-chloro-2,3,4,5-tetrahydro-1R-methyl-1H-3-benzazepine, monohydrochloride

供应商

开曼生物

产品货号

15521-50

产品报价

￥1/50mg

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产品新闻

背景资料

Lorcaserin is a full agonist of serotonin 5-HT2C receptors (Ki = 15 and 29 nM for human and rat, respectively).{25376} In functional assays it demonstrates 18- and 104-fold selectivity over 5-HT2A and 5-HT2B receptors, respectively.{25376} Chronic daily treatment with lorcaserin (ED50 = 18 mg/kg, 6 hours post dosing) has been reported to reduce food intake and body weight gain in rodents fed a high fat diet.{25376,18222} Before approving it for use in the treatment of obesity, the FDA has classified lorcaserin as a Schedule IV controlled substance.{25375}

产品描述

A selective, full agonist of serotonin 5-HT2C receptors (Ki = 15 and 29 nM for human and rat, respectively); chronic daily treatment (ED50 = 18 mg/kg, 6 hours post dosing) reduces food intake and body weight gain in rodents fed a high fat diet

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